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Molecular mechanism of regulation of the atypical protein kinase C by N-terminal domains and an allosteric small compound.
Chem Biol. 2014 Jun 19;21(6):754-65. doi: 10.1016/j.chembiol.2014.04.007. Epub 2014 May 15.
Chem Biol. 2014.
PMID: 24836908
Allosteric activation of the protein kinase PDK1 with low molecular weight compounds.
Engel M, Hindie V, Lopez-Garcia LA, Stroba A, Schaeffer F, Adrian I, Imig J, Idrissova L, Nastainczyk W, Zeuzem S, Alzari PM, Hartmann RW, Piiper A, Biondi RM.
Engel M, et al. Among authors: stroba a.
EMBO J. 2006 Nov 29;25(23):5469-80. doi: 10.1038/sj.emboj.7601416. Epub 2006 Nov 16.
EMBO J. 2006.
PMID: 17110931
Free PMC article.
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3,5-Diphenylpent-2-enoic acids as allosteric activators of the protein kinase PDK1: structure-activity relationships and thermodynamic characterization of binding as paradigms for PIF-binding pocket-targeting compounds.
Stroba A, Schaeffer F, Hindie V, Lopez-Garcia L, Adrian I, Fröhner W, Hartmann RW, Biondi RM, Engel M.
Stroba A, et al.
J Med Chem. 2009 Aug 13;52(15):4683-93. doi: 10.1021/jm9001499.
J Med Chem. 2009.
PMID: 19606904
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Structure and allosteric effects of low-molecular-weight activators on the protein kinase PDK1.
Hindie V, Stroba A, Zhang H, Lopez-Garcia LA, Idrissova L, Zeuzem S, Hirschberg D, Schaeffer F, Jørgensen TJ, Engel M, Alzari PM, Biondi RM.
Hindie V, et al. Among authors: stroba a.
Nat Chem Biol. 2009 Oct;5(10):758-64. doi: 10.1038/nchembio.208. Epub 2009 Aug 30.
Nat Chem Biol. 2009.
PMID: 19718043
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4-benzimidazolyl-3-phenylbutanoic acids as novel PIF-pocket-targeting allosteric inhibitors of protein kinase PKCζ.
Fröhner W, Lopez-Garcia LA, Neimanis S, Weber N, Navratil J, Maurer F, Stroba A, Zhang H, Biondi RM, Engel M.
Fröhner W, et al. Among authors: stroba a.
J Med Chem. 2011 Oct 13;54(19):6714-23. doi: 10.1021/jm2005892. Epub 2011 Sep 14.
J Med Chem. 2011.
PMID: 21863889
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Substrate-selective inhibition of protein kinase PDK1 by small compounds that bind to the PIF-pocket allosteric docking site.
Busschots K, Lopez-Garcia LA, Lammi C, Stroba A, Zeuzem S, Piiper A, Alzari PM, Neimanis S, Arencibia JM, Engel M, Schulze JO, Biondi RM.
Busschots K, et al. Among authors: stroba a.
Chem Biol. 2012 Sep 21;19(9):1152-63. doi: 10.1016/j.chembiol.2012.07.017.
Chem Biol. 2012.
PMID: 22999883
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