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Interactions between Gepotidacin and Escherichia coli Gyrase and Topoisomerase IV: Genetic and Biochemical Evidence for Well-Balanced Dual-Targeting.
ACS Infect Dis. 2024 Apr 12;10(4):1137-1151. doi: 10.1021/acsinfecdis.3c00346. Epub 2024 Mar 5.
ACS Infect Dis. 2024.
PMID: 38606465
Free PMC article.
Target-Mediated Fluoroquinolone Resistance in Neisseria gonorrhoeae: Actions of Ciprofloxacin against Gyrase and Topoisomerase IV.
Collins JA, Oviatt AA, Chan PF, Osheroff N.
Collins JA, et al. Among authors: oviatt aa.
ACS Infect Dis. 2024 Apr 12;10(4):1351-1360. doi: 10.1021/acsinfecdis.4c00041. Epub 2024 Mar 4.
ACS Infect Dis. 2024.
PMID: 38606464
Free PMC article.
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Topoisomerase II Poisons: Converting Essential Enzymes into Molecular Scissors.
Vann KR, Oviatt AA, Osheroff N.
Vann KR, et al. Among authors: oviatt aa.
Biochemistry. 2021 Jun 1;60(21):1630-1641. doi: 10.1021/acs.biochem.1c00240. Epub 2021 May 19.
Biochemistry. 2021.
PMID: 34008964
Free PMC article.
Review.
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Two-Dimensional Gel Electrophoresis to Resolve DNA Topoisomers.
Gibson EG, Oviatt AA, Osheroff N.
Gibson EG, et al. Among authors: oviatt aa.
Methods Mol Biol. 2020;2119:15-24. doi: 10.1007/978-1-0716-0323-9_2.
Methods Mol Biol. 2020.
PMID: 31989511
Free PMC article.
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Bimodal Actions of a Naphthyridone/Aminopiperidine-Based Antibacterial That Targets Gyrase and Topoisomerase IV.
Gibson EG, Oviatt AA, Cacho M, Neuman KC, Chan PF, Osheroff N.
Gibson EG, et al. Among authors: oviatt aa.
Biochemistry. 2019 Nov 5;58(44):4447-4455. doi: 10.1021/acs.biochem.9b00805. Epub 2019 Oct 28.
Biochemistry. 2019.
PMID: 31617352
Free PMC article.
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Polyamine-containing etoposide derivatives as poisons of human type II topoisomerases: Differential effects on topoisomerase IIα and IIβ.
Oviatt AA, Kuriappan JA, Minniti E, Vann KR, Onuorah P, Minarini A, De Vivo M, Osheroff N.
Oviatt AA, et al.
Bioorg Med Chem Lett. 2018 Sep 15;28(17):2961-2968. doi: 10.1016/j.bmcl.2018.07.010. Epub 2018 Jul 5.
Bioorg Med Chem Lett. 2018.
PMID: 30006062
Free PMC article.
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